Tesofensine – 500 mcg Research Tablets
Triple Reuptake Inhibitor for Laboratory Monoamine Transporter Studies
Overview
Tesofensine is a synthetic tropane-based compound studied in in vitro and preclinical lab models for its broad-spectrum inhibition of three major monoamine transporters: serotonin (SERT), dopamine (DAT), and norepinephrine (NET). Its triple reuptake inhibition profile supports investigations into synaptic signaling, neurotransmitter recycling, and neurochemical transporter dynamics.
Supplied in solid tablet form at 500 mcg per unit, this format ensures reproducibility in solubility, dose precision, and experimental batch control. This material is not approved for medical or diagnostic use.
Product Specifications
| Attribute | Details |
|---|---|
| Compound Name | Tesofensine |
| Form | Tablet (solid phase) |
| Content Per Tablet | 500 mcg |
| Quantity | 30 tablets per container |
| Purity | ≥99% (HPLC-verified) |
| Molecular Formula | C₁₇H₂₃Cl₂NO |
| Storage | 2–8 °C; store dry, dark |
| Shelf Life | 24 months (unopened, stored properly) |
Research Applications
Tesofensine is used exclusively in qualified lab settings for:
- Monoamine Transporter Occupancy Models: Study of SERT, DAT, and NET inhibition in controlled biochemical assays.
- Neurochemical Signaling Studies: Mapping modulation of neurotransmitters under reuptake-blockade conditions.
- Preclinical Appetite and Energy Balance Models: Laboratory analysis of central energy regulation pathways.
- Pharmacokinetic Comparisons: Evaluate transporter binding kinetics versus selective reuptake inhibitors.
All uses are investigational and must follow institutional research protocols.
Research Advantages
- Triple Transporter Inhibition: Supports multiplex assays targeting SERT, DAT, and NET simultaneously.
- Tablet Format for Laboratory Accuracy: Solid dosage allows for consistent measurement and solubility control in test systems.
- Ultra-High Purity: HPLC-verified ≥99% purity ensures reliability for pharmacological and neurochemical assessments.
Handling & Storage
- Store sealed in cool, dry, light-protected conditions
- Refrigeration at 2–8 °C recommended
- Avoid contact with moisture or high humidity
- Handle using aseptic technique in qualified laboratory facilities
- Use appropriate PPE during preparation and transfer
Disclaimer
This product is intended solely for laboratory research use. It is not a drug, supplement, or diagnostic agent, and has not been evaluated by the FDA. Any use outside approved research contexts is prohibited and voids all warranties.
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